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Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach: An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites

, , , , , , , , , , , und . Bioorg Med Chem, 17 (14): 5259-74 (Juli 2009)Michielan, Lisa Bolcato, Chiara Federico, Stephanie Cacciari, Barbara Bacilieri, Magdalena Klotz, Karl-Norbert Kachler, Sonja Pastorin, Giorgia Cardin, Riccardo Sperduti, Alessandro Spalluto, Giampiero Moro, Stefano Research Support, Non-U.S. Gov't England Bioorganic & medicinal chemistry Bioorg Med Chem. 2009 Jul 15;17(14):5259-74. Epub 2009 May 21..

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Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach: An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sites, , , , , , , , , und 2 andere Autor(en). Bioorg Med Chem, 17 (14): 5259-74 (Juli 2009)Michielan, Lisa Bolcato, Chiara Federico, Stephanie Cacciari, Barbara Bacilieri, Magdalena Klotz, Karl-Norbert Kachler, Sonja Pastorin, Giorgia Cardin, Riccardo Sperduti, Alessandro Spalluto, Giampiero Moro, Stefano Research Support, Non-U.S. Gov't England Bioorganic & medicinal chemistry Bioorg Med Chem. 2009 Jul 15;17(14):5259-74. Epub 2009 May 21..Linear and nonlinear 3D-QSAR approaches in tandem with ligand-based homology modeling as a computational strategy to depict the pyrazolo-triazolo-pyrimidine antagonists binding site of the human adenosine A2A receptor, , , , , , , , , und . J Chem Inf Model, 48 (2): 350-63 (Februar 2008)Michielan, Lisa Bacilieri, Magdalena Schiesaro, Andrea Bolcato, Chiara Pastorin, Giorgia Spalluto, Giampiero Cacciari, Barbara Klotz, Karl Norbet Kaseda, Chosei Moro, Stefano Research Support, Non-U.S. Gov't United States Journal of chemical information and modeling J Chem Inf Model. 2008 Feb;48(2):350-63. Epub 2008 Jan 24..Exploring potency and selectivity receptor antagonist profiles using a multilabel classification approach: the human adenosine receptors as a key study, , , , , , , , und . J Chem Inf Model, 49 (12): 2820-36 (Dezember 2009)Michielan, Lisa Stephanie, Federico Terfloth, Lothar Hristozov, Dimitar Cacciari, Barbara Klotz, Karl-Norbert Spalluto, Giampiero Gasteiger, Johann Moro, Stefano Research Support, Non-U.S. Gov't United States Journal of chemical information and modeling J Chem Inf Model. 2009 Dec;49(12):2820-36..